Roundtable Discussion: How Can We Advance GPCR Drug Discovery Through Cell-Based Screening & Structural Biology?

  • How can we best balance studying GPCRs in their native cellular environment versus using isolated or recombinant proteins?
  • Which protein sourcing and experimental system approaches optimise GPCR stability, activity, and translational relevance?
  • What structural biology strategies, including cryo-EM and NMR, are most effective for guiding rational GPCR drug design?